維奈妥拉
{{Infobox drug | image = Venetoclax.svg | image_class = skin-invert-image | width = 275 | alt = | image2 = Venetoclax.png | image_class2 = bg-transparent | alt2 = | caption = | pronounce = | tradename = 唯可來(Venclexta、Ven…
共 8 篇文章
{{Infobox drug | image = Venetoclax.svg | image_class = skin-invert-image | width = 275 | alt = | image2 = Venetoclax.png | image_class2 = bg-transparent | alt2 = | caption = | pronounce = | tradename = 唯可來(Venclexta、Ven…
{{Drugbox | drug_name = | IUPAC_name = (2R,3aR,10Z,11aS,12aR,14aR)-N-(Cyclopropylsulfonyl)-2-{[2-(4-isopropyl-1,3-thiazol-2-yl)-7-methoxy-8-methyl-4-quinolinyl]oxy}-5-methyl-4,14-dioxo-2,3,3a,4,5,6,7,8,9,11a,12,13,14,14a…
{{Infobox drug | drug_name = | INN = | Verifiedfields = changed | verifiedrevid = 444391072 | type = | image = Selexipag.svg | width = | alt = | caption = | pronounce = | tradename = Uptravi | Drugs.com = | MedlinePlus =…
{{Chembox | ImageFile = Asunaprevir.svg | IUPACName = 3-Methyl-N-{[(2-methyl-2-propanyl)oxy]carbonyl}-L-valyl-(4R)-4-[(7-chloro-4-methoxy-1-isoquinolinyl)oxy]-N-{(1R,2S)-1-[(cyclopropylsulfonyl)carbamoyl]-2-vinylcyclopro…
{{Infobox drug|drug_name=|type=|IUPAC_name=(1R,18R,20R,24S,27S,28S)-N-[(1R,2R)-2-(Difluoromethyl)-1-{[(1-methylcyclopropyl)sulfonyl]carbamoyl}cyclopropyl]-28-ethyl-13,13-difluoro-7-methoxy-24-(2-methyl-2-propanyl)-22,25-…
硫前列酮,或稱噻普酮,是一種類似前列腺素E2的物質,常用作催產劑, 亦可用於抗早孕。 作用机制 该药物对子宫平滑肌选择性较高,有较强子宫收缩作用,且作用时间较长。有较好的软化和扩张子宫颈管的作用,优于卡波前列素甲酯,肌内注射吸收迅速,经20-30分钟血药浓度达到峰值。临床用于抗早孕、扩宫颈及中期引产;还用于胎死宫内、异常妊娠的引产。与米非司酮合用,可提高早孕完全流产率。对产后宫缩乏力所致出血也有良效,一般用药后10分钟内出血停止。 參考…
{{chembox | ImageFile = Vaniprevir.svg | ImageSize = 275 | ImageAlt = | IUPACName = (1R,21S,24S)-21-tert-Butyl-N-((1R,2R)-1-{[(cyclopropylsulfonyl)amino]carbonyl}-2-ethylcyclopropyl)-16,16-dimethyl-3,19,22-trioxo-2,18-di…
磺胺醋酰(Sulfacetamide),是一种磺胺类人工合成抗菌药,主要通过局部用药治疗局部感染,也可以口服用于治疗泌尿道感染。 特性 磺胺醋酰室温下呈白色,水溶性强。磺胺醋酰的药物活性在磺胺类药物中处于较低水平。人口服后,磺胺醋酰能得到很好吸收,其半衰期大约是9小时,大约70%服用的磺胺醋酰会以未代谢状态经尿液排出。 磺胺醋酰对大部分的革兰氏阴性菌和革兰氏阳性菌有杀灭作用。磺胺醋酰杀灭细菌的机理和其他的磺胺类药物相似。细菌的正常生长依…